Palladium-catalyzed regioselective C2-arylation of 5-aminoindole

TAŞKESENLİGİL, Yunus; Lafzi, Ferruh; Kılıç, Haydar; SARAÇOĞLU, Nurullah

doi:10.1002/jhet.3724

Makale Tam Makale Uluslararası 2019

Palladium-catalyzed regioselective C2-arylation of 5-aminoindole

Yunus TAŞKESENLİGİL, Ferruh Lafzi, Haydar Kılıç, Nurullah SARAÇOĞLU

Journal of Heterocyclic Chemistry Cilt 56 · Sayı 12 · ss. 3289–3296 · 01.12.2019

DOI ile aç

Özet

Pd(II)-catalyzed C-H arylations of 5-aminoindole using iodobenzenes as aryl source was studied. Despite pivalamide directing group at 5-position of the indole, the direct C2-arylation of the indole observed in high yields and with high regioselectivity.

Atıf için künye

TAŞKESENLİGİL, Y., Lafzi, F., Kılıç, H., & SARAÇOĞLU, N. (2019). Palladium-catalyzed regioselective C2-arylation of 5-aminoindole. Journal of Heterocyclic Chemistry, 56(12), 3289–3296. https://doi.org/10.1002/jhet.3724

BibTeX

@article{taskesenligil2019-55539,
  author = {TAŞKESENLİGİL, Yunus and Lafzi, Ferruh and Kılıç, Haydar and SARAÇOĞLU, Nurullah},
  title = {Palladium-catalyzed regioselective C2-arylation of 5-aminoindole},
  journal = {Journal of Heterocyclic Chemistry},
  year = {2019},
  volume = {56},
  number = {12},
  pages = {3289--3296},
  issn = {0022-152X},
  doi = {10.1002/jhet.3724},
  url = {https://akademik.atauni.edu.tr/yayinlar/55539-palladium-catalyzed-regioselective-c2-arylation-of-5-aminoindole}
}