language Türkçe
Journal

ARCHIV DER PHARMAZIE

27 publications · 792 citations

Publications
Title Year Author Citations
Acetylcholinesterase and Carbonic Anhydrase Inhibition Profiles of New 5-HMF Chalcones and Their Ester Derivatives
2026 Ilhan, Ayse, Gunes, Ferhat, Erturk, Adem +3 0
Quinazolin-4(3<i>H</i>)-One-Based New Glitazones as Dual Inhibitors of α-Glucosidase and Aldose Reductase: Comprehensive Approaches for Managing Diabetes Mellitus and Its Complications
2025 Tokali, Feyzi Sinan, Demir, Yeliz, Atesoglu, Seyma +2 18
Development of Potent Type V MAPK Inhibitors: Design, Synthesis, and Biological Evaluation of Benzothiazole Derivatives Targeting p38α MAPK in Breast Cancer Cells
2025 Zoatier, Bayan, Yildiztekin, K. Gizem, Alagoz, M. Abdullah +3 5
Targeting Lung Cancer: Synthesis, Characterization, Enzyme Inhibition, and Antiproliferative Activity of 1<i>H</i>-Benzo[<i>f</i>]chromen-1-One-Thiosemicarbazones Supported by Molecular Docking
2025 Raza, Shahid, Islam, Muhammad, Cakir, Furkan +10 1
5(6)-Benzoyl-Substituted Benzimidazoles and Their Benzimidazolium Salts: Design, Synthesis, Characterization, Crystal Structure, and Some Metabolic Enzymes Inhibition Properties
2025 Aktas, Aydin, Ozden, Eda Mehtap, Celepci, Duygu Barut +6 0
Synthesis and biological studies of pyrimidine derivatives targeting metabolic enzymes
2024 Korkusuz, Elif, Sert, Yusuf, Arslan, Seher +5 40
Peripheral (<i>E</i>)-2-[(4-hydroxybenzylidene)-3,4-dihydronaphthalen-1(2<i>H</i>)-one)]-coordinated phthalocyanines with improved enzyme inhibition properties and photophysicochemical behaviors
2024 Gulec, Ozcan, Bilgicli, Ahmet T., Tuzun, Burak +5 17
Novel benzene sulfonamides with acetylcholinesterase and carbonic anhydrase inhibitory actions
2024 El Ati, Rafika, Oztaskin, Necla, Cagan, Ahmet +5 14
Synthesis of new phenothiazine derivatives: Molecular docking, assessment of cytotoxic activity and oxidant-antioxidant properties on PCS-201-012, HT-29, and SH-SY5Y cell lines
2024 Tan, Bensu, Kartal, Yasemin, Yesilyurt, Fatma +3 1
Synthesis, characterization, biochemical, and molecular modeling studies of carvacrol-based new thiosemicarbazide and 1,3,4-thiadiazole derivatives
2023 Alagoz, Tenzile, Caliskan, Fatma Gunes, Bilgicli, Hayriye Genc +4 12
Design, synthesis, a-glucosidase inhibition, pharmacokinetic, and cytotoxic studies of new indole-carbohydrazide-phenoxy-<i>N</i>-phenylacetamide derivatives
2023 Hamedifar, Haleh, Mohammadi-Khanaposhtani, Maryam, Sherafati, Maedeh +11 10
Discovery of sulfadrug-pyrrole conjugates as carbonic anhydrase and acetylcholinesterase inhibitors
2022 Gumus, Mehmet, Babacan, Semsi N., Demir, Yeliz +3 254
Some phenolic natural compounds as carbonic anhydrase inhibitors: An in vitro and in silico study
2022 Aggul, Ahmet Gokhan, Uzun, Naim, Kuzu, Muslum +2 23
Phthalimide-tethered imidazolium salts: Synthesis, characterization, enzyme inhibitory properties, and in silico studies
2022 Yigit, Murat, Demir, Yeliz, Celepci, Duygu Barut +6 14
New PEPPSI-Pd-NHC complexes bearing 4-hydroxyphenylethyl group: Synthesis, characterization, molecular docking, and bioactivity properties
2022 Behcet, Ayten, Taslimi, Parham, Gok, Yetkin +3 14
Synthesis and in vitro carbonic anhydrases and acetylcholinesterase inhibitory activities of novel imidazolinone-based benzenesulfonamides
2021 Tugrak, Mehtap, Gul, Halise Inci, Demir, Yeliz +2 66
Synthesis of novel sulfonamides with anti-Alzheimer and antioxidant capacities
2021 Gok, Nihal, Akincioglu, Akin, Binici, Edanur Erumit +3 50
Synthesis and biological evaluation of some 1-naphthol derivatives as antioxidants, acetylcholinesterase, and carbonic anhydrase inhibitors
2021 Erdogan, Musa, Kose, Leyla Polat, Essiz, Selcuk +1 46
Design, synthesis, molecular docking, and some metabolic enzyme inhibition properties of novel quinazolinone derivatives
2021 Tokali, Feyzi S., Taslimi, Parham, Demircioglu, Ibrahim H. +4 39
Synthesis of <i>N</i>-alkylated pyrazolo[3,4-<i>d</i>]pyrimidine analogs and evaluation of acetylcholinesterase and carbonic anhydrase inhibition properties
2021 Aydin, Busra O., Anil, Derya, Demir, Yeliz 39
Synthesis and in silico studies of triazene-substituted sulfamerazine derivatives as acetylcholinesterase and carbonic anhydrases inhibitors
2021 Bilginer, Sinan, Gul, Halise I., Anil, Baris +2 35
Synthesis of benzamide derivatives with thiourea-substituted benzenesulfonamides as carbonic anhydrase inhibitors
2021 Tugrak, Mehtap, Gul, Halise Inci, Demir, Yeliz +1 33
Synthesis, characterization, crystal structure, α-glycosidase, and acetylcholinesterase inhibitory properties of 1,3-disubstituted benzimidazolium salts
2021 Bal, Selma, Demirci, Ozlem, Sen, Betul +5 19
New quinoxalin-1,3,4-oxadiazole derivatives: Synthesis, characterization, in vitro biological evaluations, and molecular modeling studies
2021 Mirzazadeh, Roghieh, Asgari, Mohammad S., Barzegari, Ebrahim +10 18
A novel class for carbonic anhydrases inhibitors and evaluation of their non-zinc binding
2021 Kuzu, Burak, Tan, Meltem, Gulcin, Ilhami +1 10
Concise syntheses and some biological activities ofdl-2,5-di-<i>O</i>-methyl-<i>chiro</i>-inositol,dl-1,4-di-<i>O</i>-methyl-<i>scyllo</i>-inositol, anddl-1,6-dibromo-1,6-dideoxy-2,5-di-<i>O</i>-methyl-<i>chiro</i>-inositol
2021 Aksu, Kadir, Akincioglu, Hulya, Gulcin, Ilhami +1 9
Synthesis and biological evaluation of 3,5-diaryl-pyrazole derivatives as potential antiprostate cancer agents
2021 Anil, Derya, Caykoylu, Emine U., Sanli, Fatma +5 5